Narrow therapeutic index (NTI) medications
Therapeutic index (TI) or therapeutic ratio
The therapeutic index (TI) compares how much drug is needed to cause toxicity with how much is needed to produce the desired therapeutic effect.
It’s defined as:
TI = TD50/ED50,
where:
- TD50 is the dose that produces toxicity in 50% of the population tested.
- ED50 is the dose that produces the desired therapeutic effect in 50% of the population tested.
A higher TI generally means a safer drug, because there’s a wider gap between effective and toxic doses.
Some drugs have a narrow TI (also called NTI drugs or Narrow Therapeutic Range (NTR) drugs). With these drugs, the therapeutic and toxic doses are close together, so dosing and blood levels often need careful monitoring.